Domino allylic amination/Sonogashira/heterocyclisation reactions: palladium-catalysed three-component synthesis of pyrroles

Chem Commun (Camb). 2010 Jul 28;46(28):5157-9. doi: 10.1039/c0cc00500b. Epub 2010 Jun 7.

Abstract

Three-component reactions with 3,4-diiodoalk-2-enoic derivatives, primary amines, and terminal alkynes proceeded to give trisubstituted pyrroles in fair to good yields in the presence of palladium and copper catalysts under mild reaction conditions.

MeSH terms

  • Alkynes / chemistry
  • Amines / chemistry
  • Catalysis
  • Copper / chemistry
  • Cyclization
  • Palladium / chemistry*
  • Pyrroles / chemical synthesis*
  • Pyrroles / chemistry

Substances

  • Alkynes
  • Amines
  • Pyrroles
  • Palladium
  • Copper