Structural and functional insights into 5'-ppp RNA pattern recognition by the innate immune receptor RIG-I

Nat Struct Mol Biol. 2010 Jul;17(7):781-7. doi: 10.1038/nsmb.1863. Epub 2010 Jun 27.

Abstract

RIG-I is a cytosolic helicase that senses 5'-ppp RNA contained in negative-strand RNA viruses and triggers innate antiviral immune responses. Calorimetric binding studies established that the RIG-I C-terminal regulatory domain (CTD) binds to blunt-end double-stranded 5'-ppp RNA a factor of 17 more tightly than to its single-stranded counterpart. Here we report on the crystal structure of RIG-I CTD bound to both blunt ends of a self-complementary 5'-ppp dsRNA 12-mer, with interactions involving 5'-pp clearly visible in the complex. The structure, supported by mutation studies, defines how a lysine-rich basic cleft within the RIG-I CTD sequesters the observable 5'-pp of the bound RNA, with a stacked phenylalanine capping the terminal base pair. Key intermolecular interactions observed in the crystalline state are retained in the complex of 5'-ppp dsRNA 24-mer and full-length RIG-I under in vivo conditions, as evaluated from the impact of binding pocket RIG-I mutations and 2'-OCH(3) RNA modifications on the interferon response.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Binding Sites
  • Crystallography, X-Ray
  • DEAD Box Protein 58
  • DEAD-box RNA Helicases / chemistry*
  • DEAD-box RNA Helicases / genetics
  • DEAD-box RNA Helicases / immunology
  • DEAD-box RNA Helicases / metabolism*
  • Humans
  • Immunity, Innate
  • Interferon-Induced Helicase, IFIH1
  • Models, Molecular
  • Molecular Sequence Data
  • Nucleic Acid Conformation
  • Point Mutation
  • Protein Binding
  • Protein Conformation
  • Protein Structure, Tertiary
  • RNA Helicases / chemistry
  • RNA Helicases / metabolism
  • RNA, Double-Stranded / chemistry
  • RNA, Double-Stranded / metabolism*
  • Receptors, Immunologic
  • Sequence Alignment

Substances

  • RNA, Double-Stranded
  • Receptors, Immunologic
  • DHX58 protein, human
  • RIGI protein, human
  • IFIH1 protein, human
  • DEAD Box Protein 58
  • DEAD-box RNA Helicases
  • Interferon-Induced Helicase, IFIH1
  • RNA Helicases

Associated data

  • PDB/3NCU