Preclinical models of antipsychotic drug-induced metabolic side effects

Trends Pharmacol Sci. 2010 Oct;31(10):484-97. doi: 10.1016/j.tips.2010.07.002. Epub 2010 Aug 2.

Abstract

Antipsychotic drugs (APDs), and the 'atypical' APDs in particular, are commonly associated with metabolic side effects in humans. These include glucose dysregulation, insulin resistance, hyperlipidemia, weight gain and hypertension, which put patients at increased risk of cardiometabolic disorders. The underlying biology of APD-induced side effects in humans is poorly understood, and therefore preclinical rodent models are essential for translational research. With numerous recent studies on the topic, there is an emerging consensus that some symptoms, such as glucose dysregulation and insulin resistance, are more reliably observed than others, such as weight gain and hypertension, but, comparison between preclinical studies is complicated by numerous factors, including drug-specific effects and variables such as diet and treatment regimen. In this paper, we provide a major review of this important and growing field of preclinical study, and address crucial issues for future research.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Antipsychotic Agents / toxicity*
  • Disease Models, Animal*
  • Drug Evaluation, Preclinical / methods
  • Humans
  • Metabolic Diseases / chemically induced*
  • Metabolic Diseases / physiopathology
  • Rodentia
  • Translational Research, Biomedical / methods

Substances

  • Antipsychotic Agents