Inhibition of p38 MAPK-dependent bronchial contraction after ozone by corticosteroids

Eur Respir J. 2011 Apr;37(4):933-42. doi: 10.1183/09031936.00021110. Epub 2010 Aug 6.

Abstract

We determined the role of p38 mitogen-activated protein kinase (MAPK) in the increased airway smooth muscle (ASM) contractile responses following ozone and modulation by corticosteroids. Mice were exposed to air or ozone (3 ppm for 3 h) and isometric contractile responses of bronchial rings to acetylcholine (ACh) were measured using a myograph in the presence of p38 MAPK inhibitor, SB239063 (10⁻⁶ M) or dexamethasone (10⁻⁶ M). Because MAPK phosphatase (MKP)-1 is a negative regulator of p38 MAPK, we also studied these effects in MKP-1(-/-) mice. Bronchial rings from ozone-exposed wild-type and MKP-1(-/-) mice showed increased contractile responses, with a leftward shift of the dose-response curve in MKP-1(-/-) mice. SB239063 inhibited bronchial contraction equally in air- and ozone-exposed C57/BL6 and MKP-1(-/-) mice. Dexamethasone inhibited ACh-induced bronchial contraction in both air- and ozone-exposed C57/BL6 mice, but not in air- or ozone-exposed MKP-1(-/-) mice. ACh-stimulated p38 MAPK and heat shock protein (HSP)27 phosphorylation, as measured by Western blotting, and this effect was suppressed by SB239063 in C57/BL6 and MKP-1(-/-) mice, but not by dexamethasone in either air- or ozone-exposed MKP-1(-/-) mice. p38 MAPK plays a role in maximal ACh-induced isometric contractile responses and increased contractility induced by ozone. Dexamethasone inhibits ACh-induced ASM contraction through phosphorylation of p38 MAPK and HSP27.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylcholine / pharmacology
  • Adrenal Cortex Hormones / pharmacology*
  • Animals
  • Bronchi / drug effects
  • Bronchi / pathology*
  • Dexamethasone / pharmacology
  • Dual Specificity Phosphatase 1 / genetics
  • HSP27 Heat-Shock Proteins / metabolism
  • Humans
  • Imidazoles / pharmacology
  • Isometric Contraction
  • MAP Kinase Signaling System
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Muscle, Smooth / metabolism
  • Ozone / pharmacology*
  • Phosphorylation
  • Pyrimidines / pharmacology
  • p38 Mitogen-Activated Protein Kinases / antagonists & inhibitors*

Substances

  • Adrenal Cortex Hormones
  • HSP27 Heat-Shock Proteins
  • Imidazoles
  • Pyrimidines
  • Ozone
  • Dexamethasone
  • p38 Mitogen-Activated Protein Kinases
  • Dual Specificity Phosphatase 1
  • Dusp1 protein, mouse
  • SB 239063
  • Acetylcholine