[Everted intestinal sac method for quick finding absorption ingredients of Wuzhuyu decoction]

Zhongguo Zhong Yao Za Zhi. 2010 Jun;35(11):1399-404.
[Article in Chinese]

Abstract

Objective: To establish a method for quick finding the absorption ingredients of Wuzhuyu decoction in order to select the index to control its quality.

Method: The absorption of three concentration of Wuzhuyu decotion was investigated with the in vitro-everted intestinal sac model. The intestinal bag fluid of jejunum and ileum were collected in different time and the eight ingredients, which were evodiamine (Ev), rutaecarpine (Ru), limonin (Li), ginsenoside-Rb1, -Rg1, -Re (Rb1, Rg1, Re), isorhamnetin-3-O-beta-D-glucosyl(6''-->1'")-alpha-L-rhamnoside (Irs)and 6-gingerol (6-Gi), were detected by HPLC as the represent constituents in samples.

Result: Eight ingredients except Ru in samples could be detected, but Ev could not be detected in high concentration samples. The ratios between absorption ingredients were different from in Wuzhuyu decotion.

Conclusion: The in vitro-everted intestinal sac canc absorb the ingredients of Wuzhuyu decotion selectivity. Compare with the ileum, the jejunum can provide the more absorption information and faster, the best test time is 60-90 min.

Publication types

  • Evaluation Study

MeSH terms

  • Animals
  • Drug Evaluation, Preclinical / methods*
  • Drugs, Chinese Herbal / analysis*
  • Drugs, Chinese Herbal / pharmacokinetics*
  • Extracellular Fluid / chemistry*
  • Extracellular Fluid / drug effects
  • Ileum / chemistry
  • Ileum / drug effects
  • Intestinal Absorption*
  • Jejunum / chemistry
  • Jejunum / drug effects
  • Male
  • Rats
  • Rats, Wistar

Substances

  • Drugs, Chinese Herbal