Improved Cope-type hydroamination reactivity of hydrazine derivatives

Chem Commun (Camb). 2011 Jan 7;47(1):562-4. doi: 10.1039/c0cc02403a. Epub 2010 Oct 6.

Abstract

A systematic investigation on the metal-free, Cope-type hydroamination reactivity of hydrazides and analogues is reported. Optimization of the hydrazide structure resulted in more facile intramolecular reactivity and enabled intermolecular reactions of alkenes, thus providing a direct approach to polysubstituted hydrazides.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amination
  • Hydrazines / chemical synthesis*
  • Hydrazines / chemistry
  • Molecular Structure
  • Stereoisomerism

Substances

  • Hydrazines