The effect of doxycycline temperature-sensitive hydrogel on inhibiting the corneal neovascularization induced by BFGF in rats

Graefes Arch Clin Exp Ophthalmol. 2011 Mar;249(3):421-7. doi: 10.1007/s00417-010-1539-y. Epub 2010 Oct 16.

Abstract

Background: To study the effect of doxycycline temperature-sensitive hydrogel (DTSH) on inhibiting the corneal neovascularization (NV) induced by the basic fibroblast growth factor (bFGF).

Methods: Corneal NV was induced by slow-release polymer pellets containing bFGF, using a rat corneal pocket model. After being implanted with bFGF pellets, the female Sprague-Dawley rats were randomly divided into seven groups (12 rats/group). The grouped rats were given topically normal saline solution and neutralized DTSH at a concentration of 0%, 0.01%, 0.05%, 0.1%, 0.5%, and 1% respectively, and treated for 6 consecutive days. After 6 days of treatment, the cornea was perfused with India ink. The length and area of the corneal vessel were measured and analyzed by Image Pro-Plus 5.1.

Results: Compared to the control group given saline solution, the study groups given DTSH at a concentration of 0.05%, 0.1%, 0.5%, and 1% showed significant reduction in the vessel length (respectively, 58%, 60%, 52%, and 37%) and the vessel area (respectively, 61%, 62%, 49%, and 39%) (p < 0.001). However, no such significant reduction was observed in the study group given 0.01% DTSH (p = 0.133 and 0.166 for vessel length and area respectively). Study groups given 0.05% and 0.1% DTSH showed better effects than groups given 0.01% and 1% DTSH with regard to reducing the vessel length and the vessel area (p < 0.05).

Conclusion: The study results showed that topical DTSH effectively inhibited corneal NV at the ideal concentration of 0.05% and 0.1%. Therefore, topical DTSH could be considered as an alternative treatment for the clinical management of corneal NV.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 2-Hydroxypropyl-beta-cyclodextrin
  • Administration, Topical
  • Angiogenesis Inhibitors / administration & dosage*
  • Animals
  • Corneal Neovascularization / chemically induced
  • Corneal Neovascularization / drug therapy*
  • Corneal Neovascularization / pathology
  • Disease Models, Animal*
  • Doxycycline / administration & dosage*
  • Drug Therapy, Combination
  • Enzyme Inhibitors / administration & dosage
  • Female
  • Fibroblast Growth Factor 2
  • Matrix Metalloproteinase Inhibitors
  • Poloxamer / administration & dosage*
  • Rats
  • Rats, Sprague-Dawley
  • Temperature
  • beta-Cyclodextrins / administration & dosage*

Substances

  • Angiogenesis Inhibitors
  • Enzyme Inhibitors
  • Matrix Metalloproteinase Inhibitors
  • beta-Cyclodextrins
  • Fibroblast Growth Factor 2
  • Poloxamer
  • 2-Hydroxypropyl-beta-cyclodextrin
  • Doxycycline