Selective recognition of oncogene promoter G-quadruplexes by Mg2+

Biochem Biophys Res Commun. 2010 Nov 26;402(4):614-8. doi: 10.1016/j.bbrc.2010.10.065. Epub 2010 Oct 29.

Abstract

Mg(2+) is one of the most important cations in cells, affecting the structures and functions of the proteins and nucleic acids. It should be noted that Mg(2+) is indispensable in DNA transcription, where G-quadruplex is believed to be actively involved. Therefore, it is important to investigate the influence of Mg(2+) on G-quadruplex. Here we studied the effect of Mg(2+) on G-quadruplex DNA with CD, FRET, EMSA, and PCR-stop assay. We found that various G-quadruplexes could be differentiated through simultaneous addition of both K(+) and Mg(2+), which could be used for selective identification of G-quadruplexes in promoter oncogene but not in telomere. Mg(2+) at physiological relevant concentration not only greatly enhanced the thermostability of oncogene G-quadruplexes but also efficiently protected them from unfolding by their complementary strands, which revealed the great impact of Mg(2+) on the equilibrium between promoter G-quadruplex and duplex DNA. The PCR-stop assay further confirmed that Mg(2+) could affect gene transcription by stabilizing promoter G-quadruplex. The above studies were carried out for various G-quadruplexes of varying sequences in promoter oncogenes and telomeric region. Our results suggest that Mg(2+) may be a key regulator for G-quadruplexes of oncogene promoter, which can subsequently affect the expression of related genes.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Base Sequence
  • Circular Dichroism
  • DNA / chemistry
  • DNA / metabolism
  • Electrophoretic Mobility Shift Assay
  • Fluorescence Resonance Energy Transfer
  • G-Quadruplexes*
  • Gene Expression Regulation, Neoplastic*
  • Humans
  • Magnesium / metabolism*
  • Magnesium / pharmacology
  • Oncogenes*
  • Promoter Regions, Genetic*

Substances

  • DNA
  • Magnesium