Synthesis and preliminary pharmacological assessment of novel gamma-hydroxybutyric acid derivatives

Pol J Pharmacol Pharm. 1990 Sep-Oct;42(5):491-500.

Abstract

Synthesis and properties of new N-substituted amides of alpha-(1,1-ethylenedioxy)-ethyl-gamma-hydroxybutyric acid are described. The compounds were obtained by aminolysis of 3-(1,1-ethylenedioxy)-ethyltetra-hydrofuran-2-on with primary alkylarylamines. Preliminary pharmacological assessment revealed that the compounds exert weaker influence on the central nervous system than the reference gamma-hydroxybutyric acid. Three of the novel compounds offered some protection against pentetrazole-induced tonic seizures in mice.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Analgesics / chemical synthesis*
  • Analgesics / pharmacology
  • Animals
  • Chemical Phenomena
  • Chemistry
  • Male
  • Mice
  • Motor Activity / drug effects
  • Pentylenetetrazole / antagonists & inhibitors
  • Rats
  • Rats, Inbred Strains
  • Sodium Oxybate / analogs & derivatives*

Substances

  • Analgesics
  • Sodium Oxybate
  • Pentylenetetrazole