Biocompatibility and physicochemical characteristics of alginate-polycation microcapsules

Acta Biomater. 2011 Apr;7(4):1683-92. doi: 10.1016/j.actbio.2010.12.006. Epub 2010 Dec 8.

Abstract

There is a need for better understanding of the biocompatibility of alginate-polycation microcapsules based on their physicochemical characteristics. Microcapsules composed of alginate with 44% (IntG) or 71% (HiG) guluronate, gelled with calcium (Ca) or barium (Ba) and coated with poly-L-lysine (PLL) or poly-l-ornithine (PLO), followed by IntG alginate were compared. For microcapsules with an IntG(Ca) gel core, using PLO instead of PLL resulted in less immune cell adhesion after 2 days in C57BL/6J mice. The PLO microcapsules were also characterized by greater hydrophilicity and superior resistance to swelling and damage under osmotic stress. For microcapsules with a PLL membrane, replacing the IntG(Ca) gel core with IntG(Ba) or HiG(Ca) gel resulted in stronger immune responses (p<0.05). This was explained by poor penetration of PLL into the gel, as demonstrated by Fourier transform infrared spectroscopy analyses and membrane rupturing during osmotic swelling. X-ray photoelectron spectroscopy analyses show that all microcapsules had the same amount of polycation at their surface. Moreover, alginate coatings had non-significant effects on the biocompatibility and physicochemical properties of the microcapsules. Thus, alginate-polycation interactions for membrane formation are more important for biocompatibility than either the quantity of polycation at the surface or the alginate coating.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alginates / chemistry*
  • Alginates / pharmacology*
  • Animals
  • Biocompatible Materials / chemistry
  • Biocompatible Materials / pharmacology*
  • Capsules
  • Chemical Phenomena / drug effects*
  • Glucuronic Acid / chemistry
  • Glucuronic Acid / pharmacology
  • Hexuronic Acids / chemistry
  • Hexuronic Acids / pharmacology
  • Hydrophobic and Hydrophilic Interactions / drug effects
  • Male
  • Materials Testing / methods*
  • Membranes, Artificial
  • Mice
  • Mice, Inbred C57BL
  • Peritoneal Cavity
  • Polyamines / chemistry*
  • Polyamines / pharmacology*
  • Polyelectrolytes
  • Spectroscopy, Fourier Transform Infrared
  • Wettability / drug effects

Substances

  • Alginates
  • Biocompatible Materials
  • Capsules
  • Hexuronic Acids
  • Membranes, Artificial
  • Polyamines
  • Polyelectrolytes
  • polycations
  • Glucuronic Acid