Maternal methadone dose, placental methadone concentrations, and neonatal outcomes

Clin Chem. 2011 Mar;57(3):449-58. doi: 10.1373/clinchem.2010.154864. Epub 2011 Jan 18.

Abstract

Background: Few investigations have used placenta as an alternative matrix to detect in utero drug exposure, despite its availability at the time of birth and the large amount of sample. Methadone-maintained opioid-dependent pregnant women provide a unique opportunity to examine the placental disposition of methadone and metabolite [2-ethylidene-1,5-dimethyl-3,3-diphenylpyrrolidine (EDDP)], to explore their correlations with maternal methadone dose and neonatal outcomes, and to test the ability to detect in utero exposure to illicit drugs.

Methods: We calculated the correlations of placental methadone and EDDP concentrations and their correlations with maternal methadone doses and neonatal outcomes. Cocaine- and opiate-positive placenta results were compared with the results for meconium samples and for urine samples collected throughout gestation.

Results: Positive correlations were found between placental methadone and EDDP concentrations (r=0.685), and between methadone concentration and methadone dose at delivery (r=0.542), mean daily dose (r=0.554), mean third-trimester dose (r=0.591), and cumulative daily dose (r=0.639). The EDDP/methadone concentration ratio was negatively correlated with cumulative daily dose (r=-0.541) and positively correlated with peak neonatal abstinence syndrome (NAS) score (r=0.513). Placental EDDP concentration was negatively correlated with newborn head circumference (r=-0.579). Cocaine and opiate use was detected in far fewer placenta samples than in thrice-weekly urine and meconium samples, a result suggesting a short detection window for placenta.

Conclusions: Quantitative methadone and EDDP measurement may predict NAS severity. The placenta reflects in utero drug exposure for a shorter time than meconium but may be useful when meconium is unavailable or if documentation of recent exposure is needed.

Publication types

  • Clinical Trial
  • Research Support, N.I.H., Extramural
  • Research Support, N.I.H., Intramural

MeSH terms

  • Analgesics, Opioid / urine
  • Apgar Score
  • Birth Weight / drug effects
  • Body Size / drug effects
  • Cephalometry
  • Cocaine / urine
  • Female
  • Gestational Age
  • Humans
  • Infant, Newborn
  • Maternal Exposure* / adverse effects
  • Meconium / chemistry
  • Methadone / administration & dosage*
  • Methadone / pharmacokinetics
  • Methadone / therapeutic use
  • Opiate Substitution Treatment / methods*
  • Opioid-Related Disorders / metabolism*
  • Opioid-Related Disorders / rehabilitation
  • Opioid-Related Disorders / urine
  • Placenta / metabolism*
  • Pregnancy
  • Pregnancy Complications / metabolism*
  • Pregnancy Complications / rehabilitation
  • Pregnancy Complications / urine
  • Pregnancy Outcome
  • Pregnancy Trimesters
  • Pyrrolidines / metabolism
  • Tissue Distribution

Substances

  • Analgesics, Opioid
  • Pyrrolidines
  • Cocaine
  • Methadone
  • 2-ethylidene-1,5-dimethyl-3,3-diphenylpyrrolidine