Open vessel and cooling while heating microwave-assisted synthesis of pyridinyl N-aryl hydrazones

ACS Comb Sci. 2011 Jan 10;13(1):2-6. doi: 10.1021/co100015b. Epub 2010 Nov 9.

Abstract

We reported the first example of open vessel and cooling while heating microwave-assisted synthesis of pyridinyl N-aryl hydrazones. Compounds were prepared in excellent isolated yields (88-98%) in only 5 min, by reacting 4- and 2,4-(di)substituted phenylhydrazines, bearing both electron-donating (4-CH₃, 4-OCH₃) and -withdrawing (4-Cl, 4-Br, 4-CF₃, 4-NO₂, 2,4-Cl₂) groups with 2-, 3-, and 4-acetylpyridine. The method was successfully extended to other carbonyl compounds.

Publication types

  • Letter
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Hydrazones / chemical synthesis*
  • Hydrazones / chemistry
  • Microwaves*
  • Pyridines / chemistry*

Substances

  • Hydrazones
  • Pyridines