A novel α-isocyanoacetamide-based three-component reaction for the synthesis of dialkyl 2-acyl-5-aminofuran-3,4-dicarboxylates

Org Biomol Chem. 2011 Mar 7;9(5):1627-31. doi: 10.1039/c0ob00979b. Epub 2011 Jan 20.

Abstract

α-Isocyanoacetamides, acyl chlorides and dialkylacetylenedicarboxylates undergo a smooth multicomponent reaction to produce dialkyl 2-acyl-5-aminofuran-3,4-dicarboxylates in good yield. The scope and mechanism of this new multicomponent transformation are discussed.

MeSH terms

  • Acylation
  • Alkylation
  • Amines / chemistry*
  • Carboxylic Acids / chemical synthesis*
  • Furans / chemistry*
  • Molecular Structure
  • Nitriles / chemistry*

Substances

  • Amines
  • Carboxylic Acids
  • Furans
  • Nitriles
  • furan
  • 2-cyanoacetamide