[Effects of enalapril on NF-kappaB expression in mucus hypersecretion rats induced by acrolein exposure]

Sichuan Da Xue Xue Bao Yi Xue Ban. 2010 Nov;41(6):998-1002.
[Article in Chinese]

Abstract

Objective: To investigate the effects of enalapril on nuclear factor-kappa B (NF-kappaB) expression in a rat model of mucus hypersecretion induced by acrolein.

Methods: The rat model of mucus hypersecretion was established by the inhalation of acrolein. Then the mucus hypersecretion rats were treated by enalapril. The AB/PAS stain was performed to measure the secretion of airway in the rats, while the mRNA and protein expression levels of NF-kappaB in the airway were detected by RT-PCR, ISH, immunohistochemistry and Western blot.

Results: With the inhalation of acrolein, the airway secretion increased obviously, while the mRNA and protein expressions of NF-kappaB in lung were increased. The treatment of enalapril resulted in a significant decrease of airway secretion, as well as the downregulation of NF-kappaB in both protein and gene level.

Conclusion: Enalapril (ACE inhibitor) treatment could effectively decrease pulmonary mucus hypersecretion in acrolein-treated rats, which may be related to the downregulation of NF-kappaB expression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acrolein / toxicity*
  • Angiotensin-Converting Enzyme Inhibitors / pharmacology
  • Angiotensin-Converting Enzyme Inhibitors / therapeutic use
  • Animals
  • Enalapril / pharmacology
  • Enalapril / therapeutic use*
  • Environmental Exposure / adverse effects
  • Lung / metabolism
  • Lung Diseases / chemically induced
  • Lung Diseases / drug therapy*
  • Lung Diseases / metabolism*
  • Male
  • Mucus / metabolism
  • NF-kappa B / genetics
  • NF-kappa B / metabolism*
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Random Allocation
  • Rats
  • Rats, Sprague-Dawley

Substances

  • Angiotensin-Converting Enzyme Inhibitors
  • NF-kappa B
  • RNA, Messenger
  • Enalapril
  • Acrolein