Efficacy and safety of mizoribine combined with losartan in the treatment of IgA nephropathy: a multicenter, randomized, controlled study

Am J Med Sci. 2011 May;341(5):367-72. doi: 10.1097/MAJ.0b013e318207e02d.

Abstract

Introduction: Few have tried to prove the effectiveness of mizoribine combined with losartan for adult IgA nephropathy patients in a randomized controlled trial.

Methods: A multicenter, randomized, controlled, 12-month study was performed to evaluated the efficacy and safety of mizoribine combined with losartan for adult IgA nephropathy. Ninety-nine patients with primary IgA nephropathy from 8 clinical institutions were randomly assigned to the losartan group (n = 30), the mizoribine group (n = 35) or the combination (losartan+mizoribine) group (n = 34). The primary outcome was 24-hour urinary protein excretion (24 hours-UP).

Results: There were no significant differences in baseline data among the 3 groups. In all 3 groups, 24 hours-UP after 3, 6, 9 and 12 months of treatment were significantly lower than the baseline level. The reduction in 24 hours-UP in the losartan group was observed early and reached maximum after 6 months of treatment. Twenty-four hours-UP in the mizoribine group and combination group continuously decreased during the study. Comparisons among the 3 groups showed that the losartan group was superior to the mizoribine group after 3 months of treatment, but that after 12 months of treatment, both the combination group and the mizoribine group were superior to the losartan group in the reduction of 24 hours-UP. There were no significant differences among the 3 groups in serum creatinine. No serious adverse events occurred in any of the 3 groups.

Conclusions: The treatment of adult IgA nephropathy with mizoribine alone, losartan alone or a combination of the 2 reduced 24 hours-UP. Mizoribine and losartan, when used in combination, complement each other's activities.

Publication types

  • Multicenter Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Angiotensin Receptor Antagonists / adverse effects
  • Angiotensin Receptor Antagonists / pharmacology
  • Angiotensin Receptor Antagonists / therapeutic use*
  • Blood Pressure / drug effects
  • China
  • Creatinine / blood
  • Drug Synergism
  • Drug Therapy, Combination
  • Female
  • Glomerular Filtration Rate / drug effects
  • Glomerulonephritis, IGA / drug therapy*
  • Glomerulonephritis, IGA / metabolism
  • Humans
  • Immunosuppressive Agents / adverse effects
  • Immunosuppressive Agents / pharmacology
  • Immunosuppressive Agents / therapeutic use*
  • Longitudinal Studies
  • Losartan / adverse effects
  • Losartan / pharmacology
  • Losartan / therapeutic use*
  • Male
  • Prospective Studies
  • Proteinuria / metabolism
  • Ribonucleosides / adverse effects
  • Ribonucleosides / pharmacology
  • Ribonucleosides / therapeutic use*
  • Treatment Outcome
  • Uric Acid / blood

Substances

  • Angiotensin Receptor Antagonists
  • Immunosuppressive Agents
  • Ribonucleosides
  • Uric Acid
  • mizoribine
  • Creatinine
  • Losartan