Phosphodiesterase 5 inhibitors attenuate renal tubular apoptosis after partial unilateral ureteral obstruction: an experimental study

Kaohsiung J Med Sci. 2011 Jan;27(1):15-9. doi: 10.1016/j.kjms.2010.03.001. Epub 2011 Jan 28.

Abstract

The aim of the present study was to evaluate the effects of phosphodiesterase 5 inhibitors on renal tubular apoptosis and also on expressions of endothelial and inducible nitric oxide synthases (eNOS and iNOS) in the ipsilateral kidney after partial unilateral ureteral obstruction (PUUO) in a rat model. Forty Wistar albino rats were divided into five groups. In Groups 1-4, left experimental PUUO was created. Sildenafil, vardenafil, and tadalafil were administrated to the rats of Groups 2-4, respectively. The pills were orally given to the rats for 30 days. Group 5 was defined as sham. After 30 days, all rats were sacrificed, and nephrectomy was performed. The renal specimens were examined histopathologically. Left hydroureteronephrosis was observed in Groups 1-4. Mean apoptotic cell count and eNOS and iNOS levels were significantly increased in Group 1 when compared with the other groups. The rats in Groups 2-4 showed significantly decreased apoptotic cell count and eNOS and iNOS values in the renal tubular tissue in accordance with Group 1 (p<0.05). There were significant differences in apoptotic cell counts between sildenafil group and the other two study groups. The sildenafil group demonstrated lesser apoptotic cell count than the vardenafil (p=0.021) and tadalafil (p=0.009) groups. PUUO increases the renal tubular apoptosis and elevates NOS concentrations in renal tubular tissue after PUUO. Phosphodiesterase 5 inhibitors have a protective effect against the tubular apoptosis.

MeSH terms

  • Animals
  • Apoptosis / drug effects
  • Carbolines / pharmacology
  • Ceftriaxone / pharmacology
  • Imidazoles / pharmacology
  • Kidney Tubules / cytology*
  • Kidney Tubules / drug effects
  • Nitric Oxide Synthase Type II / metabolism
  • Nitric Oxide Synthase Type III / metabolism
  • Phosphodiesterase 5 Inhibitors / pharmacology*
  • Piperazines / pharmacology
  • Purines / pharmacology
  • Rats
  • Rats, Wistar
  • Sildenafil Citrate
  • Sulfones / pharmacology
  • Tadalafil
  • Triazines / pharmacology
  • Ureteral Obstruction*
  • Vardenafil Dihydrochloride

Substances

  • Carbolines
  • Imidazoles
  • Phosphodiesterase 5 Inhibitors
  • Piperazines
  • Purines
  • Sulfones
  • Triazines
  • Vardenafil Dihydrochloride
  • Tadalafil
  • Ceftriaxone
  • Sildenafil Citrate
  • Nitric Oxide Synthase Type II
  • Nitric Oxide Synthase Type III