Intraventricular administration of neuropeptide S has reward-like effects

Eur J Pharmacol. 2011 May 1;658(1):16-21. doi: 10.1016/j.ejphar.2011.02.009. Epub 2011 Feb 22.

Abstract

Neuropeptide S (NPS) is an endogenous brain peptide produced by neurons located in the lower brainstem, and functional studies suggest that NPS has arousing effects. Because its receptors are found in reward-associated regions throughout the brain, we evaluated whether intraventricular NPS injections elicit reward-related effects in rats. Rats increased lever presses that led to intraventricular administration of NPS (0.34-34 pmol per infusion) in a dose dependent manner, with a cue-assisted procedure. Cue-assisted self-administration of NPS was decreased by systemic administration of the dopamine receptor antagonist SCH 23390 (0.025 mg/kg, i.p.) or the hypocretin-1 (orexin-1) receptor antagonist SB 334867 (20 mg/kg, i.p.). In addition, intraventricular NPS injections (1000 pmol) induced conditioned place preference, whereas a lower dose (100 pmol) of NPS induced conditioned place aversion. Finally, NPS injections (100-1000 pmol) acutely facilitated locomotor activity, whereas repeated NPS injections did not lead to locomotor sensitization. Our data suggest that intraventricular NPS injections have reward-like effects in that NPS weakly facilitates seeking and induces positive reinforcement. These effects may depend on intact dopamine and hypocretin systems.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, N.I.H., Intramural

MeSH terms

  • Animals
  • Behavior, Animal / drug effects
  • Behavior, Animal / physiology
  • Benzazepines / pharmacology
  • Benzoxazoles / pharmacology
  • Conditioning, Psychological / drug effects
  • Conditioning, Psychological / physiology
  • Dopamine Antagonists / pharmacology
  • Injections, Intraventricular
  • Locomotion / drug effects
  • Locomotion / physiology
  • Male
  • Naphthyridines
  • Neuropeptides / administration & dosage*
  • Neuropeptides / pharmacology*
  • Rats
  • Rats, Wistar
  • Receptors, Dopamine / metabolism
  • Receptors, Neuropeptide / antagonists & inhibitors
  • Reward*
  • Self Administration
  • Urea / analogs & derivatives
  • Urea / pharmacology

Substances

  • 1-(2-methylbenzoxazol-6-yl)-3-(1,5)naphthyridin-4-yl urea
  • Benzazepines
  • Benzoxazoles
  • Dopamine Antagonists
  • Naphthyridines
  • Neuropeptides
  • Receptors, Dopamine
  • Receptors, Neuropeptide
  • SCH 23390
  • Urea