Abstract
EMBO J 30 8, 1433–1443 (2011); published online February 08 2011
In this issue of The EMBO Journal, Tanneberger et al demonstrate that Amer1/WTX, a tumour suppressor protein previously known for promoting β-catenin degradation and thus antagonizing Wnt signalling, is also required for LRP6 receptor phosphorylation and therefore activation of Wnt signalling. Amer1/WTX is recruited by PtdIns(4,5)P2 to the plasma membrane, and in turn recruits the Axin–GSK3 complex and CK1γ to phosphorylate LRP6. While dichotomic players like Amer1/WTX are common in Wnt signalling, these new findings add more intrigues to this enigmatic protein and pathway.
MeSH terms
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Adaptor Proteins, Signal Transducing
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Humans
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LDL-Receptor Related Proteins / genetics
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LDL-Receptor Related Proteins / metabolism*
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Low Density Lipoprotein Receptor-Related Protein-6
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Membrane Proteins / genetics
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Membrane Proteins / metabolism*
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Phosphatidylinositol 4,5-Diphosphate / metabolism*
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Phosphorylation
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Signal Transduction*
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Tumor Suppressor Proteins
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Wnt Proteins / genetics
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Wnt Proteins / metabolism*
Substances
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AMER1 protein, human
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Adaptor Proteins, Signal Transducing
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LDL-Receptor Related Proteins
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LRP6 protein, human
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Low Density Lipoprotein Receptor-Related Protein-6
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Membrane Proteins
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Phosphatidylinositol 4,5-Diphosphate
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Tumor Suppressor Proteins
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Wnt Proteins