Enantioselective α-amination of branched aldehydes promoted by simple chiral primary amino acids

J Org Chem. 2011 Jun 3;76(11):4661-4. doi: 10.1021/jo102361h. Epub 2011 May 6.

Abstract

A series of simple chiral primary amino acids were first successfully applied to promote the enantioselective α-amination of branched aldehydes with azadicarboxylates and the desired adducts bearing quaternary stereogenic centers were obtained in excellent yields (up to 99%) and enantioselectivities (up to 97% ee).

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aldehydes / chemistry*
  • Amination
  • Amino Acids / chemistry*
  • Stereoisomerism
  • Substrate Specificity

Substances

  • Aldehydes
  • Amino Acids