The Nudix hydrolase CDP-chase, a CDP-choline pyrophosphatase, is an asymmetric dimer with two distinct enzymatic activities

J Bacteriol. 2011 Jul;193(13):3175-85. doi: 10.1128/JB.00089-11. Epub 2011 Apr 29.

Abstract

A Nudix enzyme from Bacillus cereus (NCBI RefSeq accession no. NP_831800) catalyzes the hydrolysis of CDP-choline to produce CMP and phosphocholine. Here, we show that in addition, the enzyme has a 3'→5' RNA exonuclease activity. The structure of the free enzyme, determined to a 1.8-Å resolution, shows that the enzyme is an asymmetric dimer. Each monomer consists of two domains, an N-terminal helical domain and a C-terminal Nudix domain. The N-terminal domain is placed relative to the C-terminal domain such as to result in an overall asymmetric arrangement with two distinct catalytic sites: one with an "enclosed" Nudix pyrophosphatase site and the other with a more open, less-defined cavity. Residues that may be important for determining the asymmetry are conserved among a group of uncharacterized Nudix enzymes from Gram-positive bacteria. Our data support a model where CDP-choline hydrolysis is catalyzed by the enclosed Nudix site and RNA exonuclease activity is catalyzed by the open site. CDP-Chase is the first identified member of a novel Nudix family in which structural asymmetry has a profound effect on the recognition of substrates.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Bacillus cereus / enzymology
  • Catalytic Domain
  • Crystallography, X-Ray
  • Cytidine Diphosphate Choline / metabolism
  • Exonucleases / chemistry*
  • Exonucleases / metabolism*
  • Microscopy, Immunoelectron
  • Models, Molecular
  • Molecular Sequence Data
  • Nudix Hydrolases
  • Protein Multimerization*
  • Protein Structure, Quaternary
  • Pyrophosphatases / chemistry*
  • Pyrophosphatases / metabolism*
  • Sequence Alignment
  • Sequence Homology, Amino Acid

Substances

  • Cytidine Diphosphate Choline
  • Exonucleases
  • Pyrophosphatases

Associated data

  • PDB/3Q1P
  • PDB/3Q4I