WNT-3A modulates articular chondrocyte phenotype by activating both canonical and noncanonical pathways

J Cell Biol. 2011 May 2;193(3):551-64. doi: 10.1083/jcb.201011051.

Abstract

Activation and disruption of Wnt/β-catenin signaling both result in cartilage breakdown via unknown mechanisms. Here we show that both WNT-3A and the Wnt inhibitor DKK1 induced de-differentiation of human articular chondrocytes through simultaneous activation of β-catenin-dependent and independent responses. WNT-3A activates both the β-catenin-dependent canonical pathway and the Ca(2+)/CaMKII noncanonical pathways, with distinct transcriptional targets. WNT-3A promotes cell proliferation and loss of expression of the chondrocyte markers COL2A1, Aggrecan, and SOX9; however, proliferation and AXIN2 up-regulation are downstream of the canonical pathway and are rescued by DKK1, whereas the loss of differentiation markers is CaMKII dependent. Finally, we showed that in chondrocytes, the Ca(2+)/CaMKII-dependent and β-catenin-dependent pathways are reciprocally inhibitory, thereby explaining why DKK1 can induce loss of differentiation through de-repression of the CaMKII pathway. We propose a novel model in which a single WNT can simultaneously activate different pathways with distinct and independent outcomes and with reciprocal regulation. This offers an opportunity for selective pharmacological targeting.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cartilage, Articular / metabolism
  • Cell Differentiation
  • Cells, Cultured
  • Chondrocytes / cytology*
  • Chondrocytes / metabolism
  • Ligands
  • Mice
  • Mice, Nude
  • Models, Biological
  • Phenotype
  • Signal Transduction
  • Swine
  • Wnt Proteins / metabolism*
  • Wnt3 Protein
  • Wnt3A Protein
  • Xenopus
  • Xenopus Proteins
  • beta Catenin / metabolism

Substances

  • Ligands
  • WNT3A protein, Xenopus
  • WNT3A protein, human
  • Wnt Proteins
  • Wnt3 Protein
  • Wnt3A Protein
  • Wnt3a protein, mouse
  • Xenopus Proteins
  • beta Catenin