Nor-binaltorphimine is a reversible, noncompetitive opioid antagonist in the mouse vas deferens with high affinity for kappa receptors in monkey brain membranes

Prog Clin Biol Res. 1990:328:65-8.
No abstract available

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Cerebral Cortex / metabolism
  • In Vitro Techniques
  • Macaca mulatta
  • Male
  • Mice
  • Mice, Inbred ICR
  • Naltrexone / analogs & derivatives*
  • Naltrexone / metabolism
  • Naltrexone / pharmacology
  • Narcotic Antagonists*
  • Receptors, Opioid / metabolism
  • Receptors, Opioid, kappa
  • Synaptosomes / metabolism
  • Vas Deferens / drug effects

Substances

  • Narcotic Antagonists
  • Receptors, Opioid
  • Receptors, Opioid, kappa
  • norbinaltorphimine
  • Naltrexone