[Molecular mechanism of protective effect of puerarin solid lipid nanoparticle on cerebral ischemia-reperfusion injury in gerbils]

Zhong Yao Cai. 2010 Dec;33(12):1900-4.
[Article in Chinese]

Abstract

Objective: To investigate the effects of puerarin solid lipid nanoparticle on fore brain ischemic-reperfusion injury in gerbils and it's mechanisms.

Methods: Gerbils were randomly divided into 4 groups: sham group, cerebral ischemia-reperfusion injury group, puerarin solid lipid nanoparticle group and puerarin injection control group. The gerbils' cerebral ischemia-reperfusion injury model was constructed with ligating bilater carotids method. The histomorphology and Bcl-2, Caspase-3 and HSP70 expressions were detected by HE dyeing and immunohistochemical method.

Results: After 24 h ischemia and reperfusion in gerbils, the level of Bcl-2 and HSP70 expressions in puerarin solid lipid nanoparticle group increased (P < 0.01) compared with the ischemic-reperfusion model group, and the level of Caspase-3 expression decreased (P < 0.01). The same results was consistent in puerarin injection control group.

Conclusions: Puerarin solid lipid nanoparticle group can protect the cerebral ischemia-reperfusion injury in gerbils, which may be related to the upregulation of Bcl-2 and HSP70 expression and downregulation of Caspase-3 expression.

Publication types

  • English Abstract
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Oral
  • Animals
  • Brain / drug effects*
  • Brain / metabolism
  • Brain / pathology
  • Brain Ischemia / drug therapy
  • Brain Ischemia / metabolism
  • Brain Ischemia / prevention & control*
  • Caspase 3 / metabolism
  • Disease Models, Animal
  • Female
  • Gerbillinae
  • HSP70 Heat-Shock Proteins / metabolism
  • Immunohistochemistry
  • Isoflavones / administration & dosage
  • Isoflavones / chemistry
  • Isoflavones / pharmacology*
  • Lipids / chemistry
  • Male
  • Nanoparticles / chemistry
  • Particle Size
  • Protective Agents / administration & dosage
  • Protective Agents / pharmacology*
  • Proto-Oncogene Proteins c-bcl-2 / metabolism
  • Pueraria / chemistry
  • Random Allocation
  • Reperfusion Injury / drug therapy
  • Reperfusion Injury / metabolism
  • Reperfusion Injury / prevention & control*

Substances

  • HSP70 Heat-Shock Proteins
  • Isoflavones
  • Lipids
  • Protective Agents
  • Proto-Oncogene Proteins c-bcl-2
  • Caspase 3
  • puerarin