Minicells: versatile vectors for targeted drug or si/shRNA cancer therapy

Curr Opin Biotechnol. 2011 Dec;22(6):909-16. doi: 10.1016/j.copbio.2011.04.008. Epub 2011 May 6.

Abstract

Effective cancer therapy continues to be a daunting challenge due mainly to considerable tumor cell heterogeneity, drug-resistance, and dose-limiting toxicity of therapeutics. Here we review a versatile nano-cellular (minicell) delivery vehicle that can be packaged with therapeutically effective concentrations of chemotherapeutic drugs, siRNAs or shRNAs and can be targeted to tumors via minicell-surface attached bispecific antibodies. A range of minicell-based therapeutics have shown highly effective tumor stabilization/regression in the murine xenograft model and in case studies in canines with late-stage endogenous tumors. Repeat intravenous dosing shows absence of toxicity or immunogenicity in both species. The minicell-based therapeutic has potential applications in personalized cancer medicine.

Publication types

  • Review

MeSH terms

  • Animals
  • Antibodies / metabolism
  • Antineoplastic Agents / administration & dosage
  • Antineoplastic Agents / therapeutic use*
  • Cells / immunology
  • Cells / metabolism
  • Drug Delivery Systems*
  • Humans
  • Neoplasms / therapy*
  • RNA, Small Interfering / administration & dosage
  • RNA, Small Interfering / therapeutic use*

Substances

  • Antibodies
  • Antineoplastic Agents
  • RNA, Small Interfering