Highly enantioselective yttrium(III)-catalyzed Friedel-Crafts alkylation of β-trichloro(trifluoro)methyl aryl enones with indoles

Chem Commun (Camb). 2011 Jul 21;47(27):7821-3. doi: 10.1039/c1cc12306h. Epub 2011 Jun 8.

Abstract

An efficient yttrium(III)-catalyzed highly enantioselective Friedel-Crafts alkylation of β-trichloro(trifluoro)methyl aryl enones is described. The reaction delivered a series of functionalized indoles with a chiral tertiary carbon center bearing a trichloro(trifluoro)methyl group in excellent results (up to 96% ee and 99% yield) under mild conditions.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alkenes / chemistry*
  • Alkylation
  • Catalysis
  • Halogenation
  • Indoles / chemistry*
  • Ketones / chemistry*
  • Stereoisomerism
  • Yttrium / chemistry*

Substances

  • Alkenes
  • Indoles
  • Ketones
  • Yttrium