Estrogen receptor β-selective phytoestrogenic formulation prevents physical and neurological changes in a preclinical model of human menopause

Menopause. 2011 Oct;18(10):1131-42. doi: 10.1097/gme.0b013e3182175b66.

Abstract

Objective: As an alternative to estrogen therapy, the efficacy of an estrogen receptor β-selective phytoestrogenic (phyto-β-SERM) formulation to regulate climacteric symptoms and decline in brain responses associated with ovarian hormone loss in menopause was assessed.

Methods: A phyto-β-SERM formulation-containing diet was compared with a commercial soy extract diet and a phytoestrogen-free base/control diet in an ovariectomized (OVX) mouse model of human menopause. Two treatment studies were conducted: (1) a 2-month study assessed the effects of experimental diets on tail skin temperature as a model of menopausal hot flashes, and (2) a 9-month study assessed the long-term impact of the diets on overall health, hair thinning/loss, spatial working memory, and associated protein expression in the hippocampus.

Results: The phyto-β-SERM diet prevented OVX-induced menopause-like changes including the rise in skin temperature, hair thinning/loss, deficit in spatial memory function, and reversed OVX-induced decline in the expression of hippocampal proteins involved in neural plasticity and β-amyloid degradation/clearance. The soy extract diet had no effect or exacerbated OVX-induced changes.

Conclusions: Overall, the phyto-β-SERM diet induced physical and neurological responses comparable with ovary-intact mice, suggesting the therapeutic potential of the phyto-β-SERM formulation for the prevention/alleviation of climacteric symptoms and decline in brain responses induced by ovarian hormone loss, which provides the basis for further work in postmenopausal women.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amyloid beta-Peptides / metabolism
  • Animals
  • Disease Models, Animal
  • Estrogen Receptor beta / agonists*
  • Female
  • Hair / drug effects
  • Hippocampus / drug effects
  • Hot Flashes / drug therapy
  • Humans
  • Memory Disorders / drug therapy
  • Memory, Short-Term / drug effects
  • Menopause / drug effects*
  • Mice
  • Mice, Inbred C57BL
  • Neuronal Plasticity / drug effects
  • Phytoestrogens / administration & dosage*

Substances

  • Amyloid beta-Peptides
  • Estrogen Receptor beta
  • Phytoestrogens