Phase IB study of the combination of docetaxel, gemcitabine, and bevacizumab in patients with advanced or recurrent soft tissue sarcoma: the Axtell regimen

Ann Oncol. 2012 Mar;23(3):785-790. doi: 10.1093/annonc/mdr299. Epub 2011 Jul 11.

Abstract

Background: To assess the response of patients with soft tissue sarcoma (STS) to the combination of docetaxel, bevacizumab, and gemcitabine. Vascular endothelial growth factor (VEGF)-A levels and expression of VEGF-A and VEGF receptors 1 and 2 were evaluated.

Patients and methods: Thirty-eight chemotherapy-naive patients with STS were enrolled. A dose-finding study for gemcitabine from 1000, 1250, then 1500 mg/m(2) was done in nine patients (three cohorts), followed by an expansion cohort of 27 patients. Dose of docetaxel was 50 mg/m(2), bevacizumab was 5 mg/kg, and gemcitabine was 1500 mg/m(2), every 2 weeks. Serum VEGF-A was measured by enzyme-linked immunosorbent assay and tissue VEGF-A and its receptors by immunohistochemistry.

Results: The median follow-up was 36 months. The overall response rate observed was 31.4%, with 5 complete and 6 partial responses, and 18 stable diseases lasting for a median of 6 months. There was no significant hematologic toxicity. The adverse events with the highest grade were attributed to bevacizumab. There was no correlation of VEGF pathway biomarkers with outcome.

Conclusions: The combination of gemcitabine, docetaxel, and bevacizumab is safe and effective in patients with STS. The most concerning adverse events were consequences of bevacizumab administration. The benefit of bevacizumab in this patient population remains unclear.

Publication types

  • Clinical Trial, Phase I
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Antibodies, Monoclonal, Humanized / administration & dosage
  • Antibodies, Monoclonal, Humanized / adverse effects
  • Antineoplastic Combined Chemotherapy Protocols / therapeutic use*
  • Bevacizumab
  • Deoxycytidine / administration & dosage
  • Deoxycytidine / adverse effects
  • Deoxycytidine / analogs & derivatives
  • Disease-Free Survival
  • Docetaxel
  • Enzyme-Linked Immunosorbent Assay
  • Female
  • Gemcitabine
  • Humans
  • Immunohistochemistry
  • Kaplan-Meier Estimate
  • Male
  • Maximum Tolerated Dose
  • Middle Aged
  • Proportional Hazards Models
  • Receptors, Vascular Endothelial Growth Factor / biosynthesis
  • Sarcoma / drug therapy*
  • Sarcoma / metabolism
  • Sarcoma / mortality
  • Soft Tissue Neoplasms / drug therapy*
  • Soft Tissue Neoplasms / metabolism
  • Soft Tissue Neoplasms / mortality
  • Taxoids / administration & dosage
  • Taxoids / adverse effects
  • Vascular Endothelial Growth Factor A / biosynthesis
  • Young Adult

Substances

  • Antibodies, Monoclonal, Humanized
  • Taxoids
  • Vascular Endothelial Growth Factor A
  • Deoxycytidine
  • Docetaxel
  • Bevacizumab
  • Receptors, Vascular Endothelial Growth Factor
  • Gemcitabine