Role of superoxide radical anion in the mechanism of apoB100 degradation induced by DHA in hepatic cells

FASEB J. 2011 Oct;25(10):3554-60. doi: 10.1096/fj.11-182725. Epub 2011 Jul 14.

Abstract

VLDL is produced by the liver. Its major protein is apoB100. Docosahexaenoic acid (DHA), a dietary polyunsaturated fatty acid (PUFA), reduces VLDL levels and is used therapeutically for hypertriglyceridemia. In model systems, DHA lowers VLDL secretion by inducing presecretory apoB100 degradation, a process dependent on PUFA-derived lipid peroxides. We hypothesized that superoxide (SO) was a major participant in DHA-induced apoB100 degradation, given its promotion of lipid peroxidation. SO levels in a model of VLDL metabolism, rat hepatoma McArdle cells, were either decreased by a mimetic of superoxide dismutase 1 (SOD1) or by overexpressing SOD1 or increased by SOD1 siRNA. ApoB100 recovery was assessed by immunoprecipitation, SO by 2-hydroxyethidine, and lipid peroxides by thiobarbituric acid reactive substances. The SOD1 mimetic or SOD1 overexpression reduced SO and inhibited apoB100 degradation in DHA-treated cells by up to 100%. Surprisingly, silencing SOD1 did not increase DHA-induced degradation, although levels of SO were higher (+44%); those of lipid peroxides were similar, and their reduction by α-tocopherol decreased degradation by 50%. SO is required for lipid peroxidation in DHA-induced apoB100 degradation, but it is the peroxide level that has a tighter relationship to the level of degradation and the regulation of VLDL production.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apolipoprotein B-100 / metabolism*
  • Cell Line, Tumor
  • Docosahexaenoic Acids / pharmacology*
  • Gene Expression Regulation, Enzymologic
  • Gene Silencing
  • Hepatocytes / drug effects
  • Hepatocytes / metabolism*
  • Lipid Peroxidation
  • Metalloporphyrins
  • Mice
  • Rats
  • Superoxide Dismutase / genetics
  • Superoxide Dismutase / metabolism
  • Superoxide Dismutase-1
  • Superoxides / metabolism*

Substances

  • Apolipoprotein B-100
  • Metalloporphyrins
  • manganese(III)-tetrakis(4-benzoic acid)porphyrin
  • Superoxides
  • Docosahexaenoic Acids
  • Sod1 protein, mouse
  • Sod1 protein, rat
  • Superoxide Dismutase
  • Superoxide Dismutase-1