Inhibiting effect of bioactive metabolites produced by mushroom cultivation on bacterial quorum sensing-regulated behaviors

Chemotherapy. 2011;57(4):292-7. doi: 10.1159/000329525. Epub 2011 Jul 21.

Abstract

Aims: This study aimed to search for novel quorum sensing (QS) inhibitors from mushroom and to analyze their inhibitory activity, with a view to their possible use in controlling detrimental infections.

Methods: The bioactive metabolites produced by mushroom cultivation were tested for their abilities to inhibit QS-regulated behavior. All mushroom strains were cultivated in potato-dextrose medium by large-scale submerged fermentation. The culture supernatant was condensed into 0.2 vol by freeze-drying. The condensed supernatant was sterilized by filtration through a 0.22-μm membrane filter and added to Chromobacterium violaceum CV026 cultures, which were used to monitor QS inhibition. Inhibitory activity was measured by quantifying violacein production using a microplate reader.

Results: The results have revealed that, of 102 mushroom strains, the bioactive metabolites produced by 14 basidiomycetes were found to inhibit violacein production, a QS-regulated behavior in C. violaceum.

Conclusions: Higher fungi can produce QS-inhibitory compounds.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-Bacterial Agents / pharmacology*
  • Basidiomycota / chemistry
  • Chromobacterium / drug effects*
  • Chromobacterium / physiology
  • Drug Evaluation, Preclinical
  • Fungi / chemistry*
  • Indoles / metabolism
  • Quorum Sensing / drug effects*
  • Quorum Sensing / physiology

Substances

  • Anti-Bacterial Agents
  • Indoles
  • violacein