Effect of ketanserin, a new blocking agent of the 5-HT2 receptor, on airway responsiveness in asthma

Allergy. 1990 Feb;45(2):151-3. doi: 10.1111/j.1398-9995.1990.tb00473.x.

Abstract

Most of the antihypertensive drugs have a liability for adverse effects in asthma. Since there are few available data on the effect of ketanserin, a new antihypertensive drug which is a type-2 serotonin receptor antagonist, on human respiratory function, we have tested whether this drug can modify bronchial hyperresponsiveness to methacholine in asthmatic patients. The protective effect of intravenous ketanserin (0.14 mg/kg) was small, but significant.

Publication types

  • Clinical Trial
  • Controlled Clinical Trial
  • Randomized Controlled Trial

MeSH terms

  • Adult
  • Asthma / drug therapy*
  • Asthma / physiopathology
  • Bronchi / drug effects*
  • Bronchi / physiopathology
  • Bronchial Provocation Tests / methods
  • Child
  • Dose-Response Relationship, Immunologic
  • Female
  • Forced Expiratory Volume
  • Humans
  • Ketanserin / pharmacology*
  • Male
  • Methacholine Chloride
  • Methacholine Compounds / administration & dosage
  • Methacholine Compounds / antagonists & inhibitors*
  • Methacholine Compounds / immunology
  • Serotonin Antagonists / pharmacology

Substances

  • Methacholine Compounds
  • Serotonin Antagonists
  • Methacholine Chloride
  • Ketanserin