Highly diastereoselective vinylogous Mukaiyama aldol reaction of α-keto phosphonates with 2-(trimethylsilyloxy)furan catalyzed by Cu(OTf)2

Org Biomol Chem. 2011 Oct 7;9(19):6721-6. doi: 10.1039/c1ob05822c. Epub 2011 Aug 4.

Abstract

The diastereospecific formation of δ-hydroxyalkylbutenolide phosphonate has been achieved via a vinylogous Mukaiyama aldol reaction. The reaction was performed using α-ketophosphonate 1 and 2-(trimethylsilyloxy)furan 2 mediated by Cu(OTf)(2) and 2,2,2-trifluoroethanol as additive in CH(2)Cl(2). The reaction proceeds rapidly and affords the corresponding 5-(hydroxy(aryl)methyl) furan-2(5H)-one phosphonates 3 in high yields with good to excellent diastereoselectivities (d.r. up to >99 : 1). 5-(Hydroxy(alkyl)methyl)furan-2(5H)-one phosphonates could also be obtained with good diastereoselectivities.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Catalysis
  • Crystallography, X-Ray
  • Furans / chemical synthesis
  • Furans / chemistry*
  • Ketones / chemistry*
  • Mesylates / chemistry*
  • Models, Molecular
  • Molecular Structure
  • Organophosphonates / chemical synthesis
  • Organophosphonates / chemistry*
  • Stereoisomerism
  • Trifluoroethanol / chemistry
  • Trimethylsilyl Compounds / chemistry*

Substances

  • Furans
  • Ketones
  • Mesylates
  • Organophosphonates
  • Trimethylsilyl Compounds
  • Trifluoroethanol
  • trifluoromethanesulfonic acid