Adipolin/C1qdc2/CTRP12 protein functions as an adipokine that improves glucose metabolism

J Biol Chem. 2011 Oct 7;286(40):34552-8. doi: 10.1074/jbc.M111.277319. Epub 2011 Aug 17.

Abstract

Obesity is a major risk factor for the development of insulin resistance and type 2 diabetes. Adipose tissue secretes various bioactive molecules, referred to as adipokines, whose dysregulation can mediate changes in glucose homeostasis and inflammatory responses. Here, we identify C1qdc2/CTRP12 as an insulin-sensitizing adipokine that is abundantly expressed by fat tissues and designate this adipokine as adipolin (adipose-derived insulin-sensitizing factor). Adipolin expression in adipose tissue and plasma was reduced in rodent models of obesity. Adipolin expression was also decreased in cultured 3T3-L1 adipocytes by treatment with inducers of endoplasmic reticulum stress and inflammation. Systemic administration of adipolin ameliorated glucose intolerance and insulin resistance in diet-induced obese mice. Adipolin administration also reduced macrophage accumulation and proinflammatory gene expression in the adipose tissue of obese mice. Conditioned medium from adipolin-expressing cells diminished the expression of proinflammatory cytokines in response to stimulation with LPS or TNFα in cultured macrophages. These data suggest that adipolin functions as an anti-inflammatory adipokine that exerts beneficial actions on glucose metabolism. Therefore, adipolin represents a new target molecule for the treatment of insulin resistance and diabetes.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3T3-L1 Cells
  • Adipokines / genetics
  • Adipokines / metabolism*
  • Adipokines / physiology
  • Animals
  • COS Cells
  • Chlorocebus aethiops
  • Cloning, Molecular
  • Endoplasmic Reticulum / metabolism
  • Glucose / metabolism*
  • Inflammation
  • Lipopolysaccharides / metabolism
  • Macrophages / metabolism
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Models, Biological
  • Obesity
  • Tumor Necrosis Factor-alpha / metabolism

Substances

  • Adipokines
  • C1qtnf12 protein, mouse
  • Lipopolysaccharides
  • Tumor Necrosis Factor-alpha
  • Glucose