Intramolecular aryne-ene reaction: synthetic and mechanistic studies

J Am Chem Soc. 2011 Sep 14;133(36):14200-3. doi: 10.1021/ja205405n. Epub 2011 Aug 19.

Abstract

Although the chemistry of arynes is well developed, some challenges still remain. The ene reaction of arynes has not gained widespread use in synthesis as a result of poor yields and selectivity. A general, high yielding and selective intramolecular aryne-ene reaction is described providing various benzofused carbo- and heterocycles. Mechanistic data is presented, and a rationale for the resulting stereochemistry is discussed.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Organic Chemicals / chemical synthesis*
  • Organic Chemicals / chemistry

Substances

  • Organic Chemicals