Tumor suppressor protein (p)53, is a regulator of NF-kappaB repression by the glucocorticoid receptor

Proc Natl Acad Sci U S A. 2011 Oct 11;108(41):17117-22. doi: 10.1073/pnas.1114420108. Epub 2011 Sep 26.

Abstract

Glucocorticoids can inhibit inflammation by abrogating the activity of NF-κB, a family of transcription factors that regulates the production of proinflammatory cytokines. To understand the molecular mechanism of repression of NF-κB activity by glucocorticoids, we performed a high-throughput siRNA oligo screen to identify novel genes involved in this process. Here, we report that loss of p53, a tumor suppressor protein, impaired repression of NF-κB target gene transcription by glucocorticoids. Additionally, loss of p53 also impaired transcription of glucocorticoid receptor (GR) target genes, whereas upstream NF-κB and glucocorticoid receptor signaling cascades remained intact. We further demonstrate that p53 loss severely impaired glucocorticoid rescue of death in a mouse model of LPS shock. Our findings unveil a new role for p53 in the repression of NF-κB by glucocorticoids and suggest important implications for treatment of the proinflammatory microenvironments found in tumors with aberrant p53 activity.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Validation Study

MeSH terms

  • Animals
  • Dexamethasone / pharmacology
  • High-Throughput Screening Assays
  • Lipopolysaccharides / toxicity
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • NF-kappa B / metabolism*
  • Protein Interaction Maps
  • RNA Interference
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • RNA, Small Interfering / genetics
  • Receptors, Glucocorticoid / metabolism*
  • Shock, Septic / chemically induced
  • Shock, Septic / genetics
  • Shock, Septic / metabolism
  • Signal Transduction
  • Tumor Suppressor Protein p53 / deficiency
  • Tumor Suppressor Protein p53 / genetics
  • Tumor Suppressor Protein p53 / metabolism*

Substances

  • Lipopolysaccharides
  • NF-kappa B
  • RNA, Messenger
  • RNA, Small Interfering
  • Receptors, Glucocorticoid
  • Tumor Suppressor Protein p53
  • Dexamethasone