Dendritic carrier based on PEG: design and degradation of acid-sensitive dendrimer-like poly(ethylene oxide)s

Macromol Rapid Commun. 2011 Nov 1;32(21):1722-8. doi: 10.1002/marc.201100459. Epub 2011 Sep 14.

Abstract

Degradable dendrimer-like PEOs were designed using an original ABC-type branching agent featuring a cleavable ketal group, following an iterative divergent approach based on the anionic ring opening polymerization (AROP) of ethylene oxide and arborization of PEO chain ends. A seventh generation dendrimer-like PEO carrying 192 peripheral hydroxyls and exhibiting a molar mass of 446 kg · mol(-1) was obtained in this way. The chemical degradation of these dendritic scaffolds was next successfully accomplished under acidic conditions, forming linear PEO chains of low molar mass (≈2 kg · mol(-1)), as monitored by (1)H NMR, SEC, and MALDI-TOF mass spectrometry as well as by AFM.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Dendrimers / chemical synthesis
  • Dendrimers / chemistry*
  • Drug Carriers / chemical synthesis
  • Drug Carriers / chemistry*
  • Drug Delivery Systems / instrumentation*
  • Molecular Weight
  • Polyethylene Glycols / chemistry*

Substances

  • Dendrimers
  • Drug Carriers
  • Polyethylene Glycols