Allelic combinations of immune-response genes associated with glatiramer acetate treatment response in Russian multiple sclerosis patients

Pharmacogenomics. 2012 Jan;13(1):43-53. doi: 10.2217/pgs.11.136. Epub 2011 Nov 23.

Abstract

Background: Glatiramer acetate (GA) is widely used as a first-line disease-modifying treatment for multiple sclerosis (MS). However, a significant proportion of MS patient appears to experience modest benefit from GA-treatment. Genetic variants affecting the clinical response to GA are believed to be relevant as biomarkers of GA-treatment efficiency.

Patients & methods: Nine polymorphisms in candidate genes were analyzed as possible determinants of GA response in 285 Russian MS patients. Special attention was given to identification of response-associated allelic combinations by means of the APSampler algorithm.

Results: No significant associations were found for individual polymorphisms. Alleles DRB1*15, TGFB1*T, CCR5*d and IFNAR1*G were the components of the combinations, of which carriage was significantly higher in nonresponders than in responders. Carriers of the most significant combinations: DRB1*15 + TGFB1*T + CCR5*d + IFNAR1*G and DRB1*15 + TGFB1*T + CCR5*d (permutation p-values: 0.0056 and 0.013, respectively) had a 14 to 15-times increased risk of ineffective response to GA therapy.

Discussion: The results suggest that the influence of immune-response genes on GA-induced response has a polygenic nature. The data are interpreted as evidence of additive and epistatic influences of the genes on GA efficiency for MS treatment.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Alleles
  • Biomarkers, Pharmacological / blood
  • Epistasis, Genetic
  • Female
  • Genes, MHC Class II / genetics
  • Genetic Association Studies
  • Glatiramer Acetate
  • HLA-DRB1 Chains / genetics*
  • Humans
  • Male
  • Middle Aged
  • Multifactorial Inheritance
  • Multiple Sclerosis / drug therapy*
  • Multiple Sclerosis / genetics
  • Peptides / therapeutic use*
  • Receptor, Interferon alpha-beta / genetics*
  • Receptors, CCR5 / genetics*
  • Transforming Growth Factor beta1 / genetics*

Substances

  • Biomarkers, Pharmacological
  • HLA-DRB1 Chains
  • IFNAR1 protein, human
  • Peptides
  • Receptors, CCR5
  • TGFB1 protein, human
  • Transforming Growth Factor beta1
  • Receptor, Interferon alpha-beta
  • Glatiramer Acetate