Clinical significance of BRAF gene mutations in patients with non-small cell lung cancer

Anticancer Res. 2011 Dec;31(12):4619-23.

Abstract

Background: V-raf murine sarcoma viral oncogene homolog B1 (BRAF) mutations are attractive molecular targets for cancer treatment. Detection of BRAF gene mutation and analyses in non-small cell lung cancer (NSCLC) are of great scientific interest.

Patients and methods: The study included 581 NSCLC patients (377 males, 204 female) undergoing pulmonary resection. BRAF gene mutations were screened using the PCR-SSCP method and were confirmed by direct DNA sequencing. Mutations of epidermal growth factor receptor (EGFR), v-erb-b2 erythroblastic leukemia viral oncogene homolog 2 (ERBB2), and v-Ki-ras2 Kirsten rat sarcoma viral oncogene homolog (KRAS) gene were also analyzed.

Results: Five patients (0.8%) had BRAF mutations within exon 15. In 581 NSCLC patients, EGFR gene mutations within exons 18 to 21 were detected in 191 (32.8%) patients, KRAS codon 12 mutations in 56 (9.6%) patients, and ERBB2 codon 20 mutations in 11 (1.8%) patients. All mutations were mutually exclusive. The NSCLC patients with BRAF mutations were proved to be men who were heavy smokers.

Conclusions: PCR-SSCP analysis of BRAF exon 15 in NSCLC patients without other gene mutations may be sufficient to identify candidates for treatment.

MeSH terms

  • Adenocarcinoma / genetics*
  • Aged
  • Carcinoma, Non-Small-Cell Lung / genetics*
  • Carcinoma, Squamous Cell / genetics*
  • Codon
  • DNA Mutational Analysis
  • Exons
  • Female
  • Gene Expression Regulation, Neoplastic*
  • Genes, erbB-2 / genetics
  • Genes, ras / genetics
  • Humans
  • Lung Neoplasms / genetics*
  • Male
  • Middle Aged
  • Mutation*
  • Polymorphism, Single-Stranded Conformational
  • Proto-Oncogene Proteins B-raf / genetics*

Substances

  • Codon
  • BRAF protein, human
  • Proto-Oncogene Proteins B-raf