Shortened Ca2+ signaling refractoriness underlies cellular arrhythmogenesis in a postinfarction model of sudden cardiac death

Circ Res. 2012 Feb 17;110(4):569-77. doi: 10.1161/CIRCRESAHA.111.260455. Epub 2012 Jan 5.

Abstract

Rationale: Diastolic spontaneous Ca(2+) waves (DCWs) are recognized as important contributors to triggered arrhythmias. DCWs are thought to arise when [Ca(2+)] in sarcoplasmic reticulum ([Ca(2+)](SR)) reaches a certain threshold level, which might be reduced in cardiac disease as a consequence of sensitization of ryanodine receptors (RyR2s) to luminal Ca(2+).

Objective: We investigated the mechanisms of DCW generation in myocytes from normal and diseased hearts, using a canine model of post-myocardial infarction ventricular fibrillation (VF).

Methods and results: The frequency of DCWs, recorded during periodic pacing in the presence of a β-adrenergic receptor agonist isoproterenol, was significantly higher in VF myocytes than in normal controls. Rather than occurring immediately on reaching a final [Ca(2+)](SR), DCWs arose with a distinct time delay after attaining steady [Ca(2+)](SR) in both experimental groups. Although the rate of [Ca(2+)](SR) recovery after the SR Ca(2+) release was similar between the groups, in VF myocytes the latency to DCWs was shorter, and the [Ca(2+)](SR) at DCW initiation was lower. The restitution of depolarization-induced Ca(2+) transients, assessed by a 2-pulse protocol, was significantly faster in VF myocytes than in controls. The VF-related alterations in myocyte Ca(2+) cycling were mimicked by the RyR2 agonist, caffeine. The reducing agent, mercaptopropionylglycine, or the CaMKII inhibitor, KN93, decreased DCW frequency and normalized restitution of Ca(2+) release in VF myocytes.

Conclusions: The attainment of a certain threshold [Ca(2+)](SR) is not sufficient for the generation of DCWs. Postrelease Ca(2+) signaling refractoriness critically influences the occurrence of DCWs. Shortened Ca(2+) signaling refractoriness due to RyR2 phosphorylation and oxidation is responsible for the increased rate of DCWs observed in VF myocytes and could provide a substrate for synchronization of arrhythmogenic events at the tissue level in hearts prone to VF.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adrenergic beta-Agonists
  • Animals
  • Benzylamines / pharmacology
  • Caffeine / pharmacology
  • Calcium Channel Agonists / pharmacology
  • Calcium Signaling* / drug effects
  • Calcium-Calmodulin-Dependent Protein Kinase Type 2 / antagonists & inhibitors
  • Calcium-Calmodulin-Dependent Protein Kinase Type 2 / metabolism
  • Cardiac Pacing, Artificial
  • Death, Sudden, Cardiac / etiology*
  • Disease Models, Animal
  • Dogs
  • Excitation Contraction Coupling
  • Female
  • Isoproterenol
  • Male
  • Myocardial Infarction / complications*
  • Myocardial Infarction / metabolism
  • Myocardial Infarction / physiopathology
  • Myocytes, Cardiac / drug effects
  • Myocytes, Cardiac / metabolism*
  • Oxidation-Reduction
  • Phosphorylation
  • Protein Kinase Inhibitors / pharmacology
  • Reaction Time
  • Reducing Agents / pharmacology
  • Ryanodine Receptor Calcium Release Channel / drug effects
  • Ryanodine Receptor Calcium Release Channel / metabolism
  • Sarcoplasmic Reticulum / metabolism
  • Sulfonamides / pharmacology
  • Time Factors
  • Tiopronin / pharmacology
  • Ventricular Fibrillation / etiology*
  • Ventricular Fibrillation / metabolism
  • Ventricular Fibrillation / physiopathology

Substances

  • Adrenergic beta-Agonists
  • Benzylamines
  • Calcium Channel Agonists
  • Protein Kinase Inhibitors
  • Reducing Agents
  • Ryanodine Receptor Calcium Release Channel
  • Sulfonamides
  • KN 93
  • Caffeine
  • Tiopronin
  • Calcium-Calmodulin-Dependent Protein Kinase Type 2
  • Isoproterenol