A new and convenient approach for the preparation of β-cyanoethyl protected trinucleotide phosphoramidites

Org Biomol Chem. 2012 Feb 28;10(8):1510-3. doi: 10.1039/c2ob06934b. Epub 2012 Jan 10.

Abstract

Herein we report a convenient approach for the preparation of fully protected trinucleotide synthons to be used for the synthesis of gene libraries. The trinucleotide synthons bear β-cyanoethyl groups at the phosphate residues, and thus can be used in standard oligonucleotide synthesis without additional steps for deprotection and work-up.

MeSH terms

  • Cyanates / chemistry*
  • Molecular Structure
  • Oligonucleotides / chemistry*
  • Organophosphorus Compounds / chemistry*
  • Phosphorylation

Substances

  • Cyanates
  • Oligonucleotides
  • Organophosphorus Compounds
  • phosphoramidite