A DR4:tBID axis drives the p53 apoptotic response by promoting oligomerization of poised BAX

EMBO J. 2012 Mar 7;31(5):1266-78. doi: 10.1038/emboj.2011.498. Epub 2012 Jan 13.

Abstract

The cellular response to p53 activation varies greatly in a stimulus- and cell type-specific manner. Dissecting the molecular mechanisms defining these cell fate choices will assist the development of effective p53-based cancer therapies and also illuminate fundamental processes by which gene networks control cellular behaviour. Using an experimental system wherein stimulus-specific p53 responses are elicited by non-genotoxic versus genotoxic agents, we discovered a novel mechanism that determines whether cells undergo proliferation arrest or cell death. Strikingly, we observe that key mediators of cell-cycle arrest (p21, 14-3-3σ) and apoptosis (PUMA, BAX) are equally activated regardless of outcome. In fact, arresting cells display strong translocation of PUMA and BAX to the mitochondria, yet fail to release cytochrome C or activate caspases. Surprisingly, the key differential events in apoptotic cells are p53-dependent activation of the DR4 death receptor pathway, caspase 8-mediated cleavage of BID, and BID-dependent activation of poised BAX at the mitochondria. These results reveal a previously unappreciated role for DR4 and the extrinsic apoptotic pathway in cell fate choice following p53 activation.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis Regulatory Proteins / metabolism
  • Apoptosis*
  • BH3 Interacting Domain Death Agonist Protein / metabolism*
  • Caspase 8 / metabolism
  • Cell Proliferation
  • Humans
  • Mitochondria / metabolism
  • Protein Transport
  • Proto-Oncogene Proteins / metabolism
  • Receptors, TNF-Related Apoptosis-Inducing Ligand / metabolism*
  • Tumor Suppressor Protein p53 / metabolism*
  • bcl-2-Associated X Protein / metabolism*

Substances

  • Apoptosis Regulatory Proteins
  • BBC3 protein, human
  • BH3 Interacting Domain Death Agonist Protein
  • Proto-Oncogene Proteins
  • Receptors, TNF-Related Apoptosis-Inducing Ligand
  • TNFRSF10A protein, human
  • Tumor Suppressor Protein p53
  • bcl-2-Associated X Protein
  • Caspase 8