Liver microsome-mediated mutagenicity of dihydrodiols derived from dibenz(a,c)anthracene in S. typhimurium TA100

Carcinogenesis. 1980 Mar;1(3):287-9. doi: 10.1093/carcin/1.3.287.

Abstract

The mutagenic activities of the trans-1,2- and 3,4-diols of dibenz(a,c)anthracene, both of which could yield 'bay-region' diol-epoxides on further metabolism, were lower than those of the parent hydrocarbon and of the related 10,11-diol.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Benz(a)Anthracenes / pharmacology*
  • Dihydroxydihydrobenzopyrenes / pharmacology*
  • Microsomes, Liver / drug effects*
  • Molecular Structure
  • Mutagenicity Tests
  • Rats
  • Salmonella typhimurium / drug effects*
  • Structure-Activity Relationship

Substances

  • Benz(a)Anthracenes
  • Dihydroxydihydrobenzopyrenes
  • benzanthracene-10,11-dihydrodiol
  • 3,4-dihydro-3,4-dihydroxybenzo(a,i)pyrene
  • 1,2-dihydro-1,2-dihydroxydibenzo(a)pyrene