The anomeric mixture of some O-galactolipid derivatives is more toxic against cancer cells than either anomer alone

Bioorg Med Chem Lett. 2012 Mar 1;22(5):2030-2. doi: 10.1016/j.bmcl.2012.01.069. Epub 2012 Jan 28.

Abstract

The anomeric mixture of a series of O-galactolipid derivatives is revealed to be more toxic against several cancer cell lines than their either single component with the pure α- or β-configuration. This interesting phenomenon has been confirmed on pairs of synthesized O-galactosyl anomers bearing length-varied alkyl chains at the lipid end. Furthermore, the most potent mixture was determined inoffensive to a normal cell line tested.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antineoplastic Agents / chemistry*
  • Antineoplastic Agents / pharmacology*
  • Cell Line, Tumor
  • Cell Survival / drug effects
  • Drug Synergism
  • Galactolipids / chemistry*
  • Galactolipids / pharmacology*
  • Humans
  • Neoplasms / drug therapy

Substances

  • Antineoplastic Agents
  • Galactolipids