The potential of laminin-2-biomimetic short peptide to promote cell adhesion, spreading and migration by inducing membrane recruitment and phosphorylation of PKCδ

Biomaterials. 2012 May;33(15):3967-79. doi: 10.1016/j.biomaterials.2012.02.002. Epub 2012 Feb 24.

Abstract

Laminin α2 chain plays an important role in basement membrane assembly and peripheral myelinogenesis; however, the integrin binding motif within human laminin α2 chain and the signaling pathways downstream of this ligand-receptor interaction are poorly understood. We identified a motif, RNIPPFEGCIWN (Ln2-LG3-P2), within LG3 domain of human laminin α2 chain as a major site for both α3β1 integrin and cellular activities such as cell adhesion, spreading, and migration. Binding of α3β1 integrin with Ln2-LG3-P2 induced the membrane recruitment of protein kinase Cδ (PKCδ) and stimulated its tyrosine phosphorylation. The cellular activities induced by Ln2-LG3-P2 and the phosphorylation of focal adhesion kinase (FAK) were inhibited by rottlerin, a PKCδ inhibitor, but not by Gö6976, a PKCα/β inhibitor. These results indicate that RNIPPFEGCIWN motif within human laminin α2 chain is a major ligand for α3β1 integrin, and that binding of α3β1 integrin mediates cellular activities through membrane recruitment and tyrosine phosphorylation of PKCδ and FAK phosphorylation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Motifs
  • Amino Acid Sequence
  • Animals
  • Arginine / metabolism
  • Biomimetic Materials / chemistry
  • Biomimetic Materials / pharmacology*
  • Cell Adhesion / drug effects
  • Cell Membrane / drug effects
  • Cell Membrane / enzymology*
  • Cell Movement / drug effects*
  • Focal Adhesion Protein-Tyrosine Kinases / metabolism
  • Focal Adhesions / drug effects
  • Focal Adhesions / metabolism
  • Humans
  • Integrin alpha3beta1 / metabolism
  • Laminin / chemistry
  • Laminin / isolation & purification
  • Laminin / pharmacology*
  • Molecular Sequence Data
  • PC12 Cells
  • Peptides / chemistry
  • Peptides / isolation & purification
  • Peptides / pharmacology*
  • Phosphorylation / drug effects
  • Phosphotyrosine / metabolism
  • Protein Binding / drug effects
  • Protein Kinase C-delta / metabolism*
  • Protein Structure, Tertiary
  • Protein Transport / drug effects
  • Rats
  • Stress Fibers / drug effects
  • Stress Fibers / metabolism

Substances

  • Integrin alpha3beta1
  • Laminin
  • Peptides
  • Phosphotyrosine
  • Arginine
  • Focal Adhesion Protein-Tyrosine Kinases
  • Protein Kinase C-delta