Antithrombotic activity of protein S infused without activated protein C in a baboon thrombosis model

Thromb Haemost. 2012 Apr;107(4):690-8. doi: 10.1160/TH11-10-0699. Epub 2012 Feb 28.

Abstract

Protein S (ProS) is an essential plasma protein that enhances the anticoagulant activity of activated protein C (APC). In vitro , purified native human Zn2+-containing ProS also exerts direct anticoagulant activity by inhibiting prothrombinase and extrinsic FXase activities independently of APC. We investigated antithrombotic effects of ProS infused without APC in a baboon shunt model of thrombogenesis that employs a device consisting of arterial and venous shear flow segments. In in vitro experiments, the Zn2+-containing human ProS used for the studies displayed >10-fold higher prothrombinase inhibitory activity and anticoagulant activity in tissue factor-stimulated plasma, and four-fold higher inhibition of the intrinsic pathway than the Zn2+-deficient ProS used. In the thrombosis model, ProS (33 μg/minute for 1 hour) or saline was infused locally; platelet and fibrin deposition in the shunt were measured over 2 hours. During experiments performed at 50 ml/minute blood flow, Zn2+-containing ProS inhibited platelet deposition 73-96% in arterial-type flow segments and 90-99% in venous-type flow segments; Zn2+-deficient ProS inhibited platelet deposition 52% in arterial-type flow segments and 65-73% in venous-type flow segments. At 100 ml/min blood flow rate, Zn2+-containing ProS inhibited platelet deposition by 39% and 73% in the respective segments; Zn2+-deficient ProS inhibited platelet deposition by 5% and 0% in the respective segments. Zn2+-containing ProS suppressed fibrin deposition by 67-90%. Systemic APC-independent ProS activity was significantly increased and thrombin-antithrombin complex levels were significantly decreased after infusion of ProS. Thus, infused human Zn2+-containing ProS is antithrombotic in primates, and may have therapeutic potential even in protein C-deficient human patients.

MeSH terms

  • Animals
  • Anticoagulants / metabolism
  • Blood Platelets / metabolism
  • Cysteine Endopeptidases / metabolism
  • Disease Models, Animal
  • Fibrin / metabolism
  • Fibrinolytic Agents / pharmacology
  • Hemostasis
  • Humans
  • Male
  • Neoplasm Proteins / metabolism
  • Papio
  • Protein C / metabolism*
  • Protein C Deficiency / metabolism
  • Protein S / metabolism*
  • Thrombosis / metabolism*
  • Thrombosis / pathology
  • Time Factors
  • Zinc / chemistry

Substances

  • Anticoagulants
  • Fibrinolytic Agents
  • Neoplasm Proteins
  • Protein C
  • Protein S
  • Fibrin
  • Cysteine Endopeptidases
  • cancer procoagulant
  • Zinc