[Choice of a spin label probe in order to study the recombination of beta-hydroxybutyrate dehydrogenase of a rat liver inner mitochondrial membrane with lecithin vesicles]

C R Seances Acad Sci D. 1979 Jan 22;288(3):363-5.
[Article in French]

Abstract

We find from studying the inhibitory effect of N-ethylmaleimide (NEM) on the enzymatic activity of beta-hydroxybutyrate dehydrogenase, that approximately one molecule of NEM is bound for one molecule of protein when the enzymatic activity is completely inhibited. Since the protein is a dimer this implies that each molecule of protein possesses only one thiol group in its catalytic center. Two long chain maleimide derivates: (10.3) NEM and (1.14) NEM conform, if a reasonable assumption is accepted to the conditions required for the study of the recombination of beta-hydroxybutyrate dehydrogenase with lecithin vesicles by spin label technique.

Publication types

  • English Abstract

MeSH terms

  • Animals
  • Binding Sites
  • Electron Spin Resonance Spectroscopy
  • Ethylmaleimide / pharmacology
  • Hydroxybutyrate Dehydrogenase / antagonists & inhibitors
  • Hydroxybutyrate Dehydrogenase / metabolism*
  • Iodoacetamide / pharmacology
  • Maleimides / chemical synthesis
  • Maleimides / pharmacology
  • Mitochondria, Liver / enzymology*
  • Phosphatidylcholines / metabolism*
  • Rats
  • Spin Labels* / chemical synthesis

Substances

  • Maleimides
  • Phosphatidylcholines
  • Spin Labels
  • Hydroxybutyrate Dehydrogenase
  • Ethylmaleimide
  • Iodoacetamide