GemAffinity: a scoring function for predicting binding affinity and virtual screening

Int J Data Min Bioinform. 2012;6(1):27-41. doi: 10.1504/ijdmb.2012.045535.

Abstract

Prediction of protein-ligand binding affinities plays an essential role for molecular recognition and virtual screening. We have developed a scoring function, namely GemAffinity, to predict binding affinities by using a stepwise regression method and 88 descriptors from 891 complex structures. GemAffinity consists of five descriptors, including van der Waals contacts; metal-ligand interactions; water effects; ligand deformation penalty; and conserved hydrogen-bonded residues. Experimental results indicate that GemAffinity is the best among 13 methods on a test set and can enrich screening accuracies on four sets. We believe that GemAffinity is useful for virtual screening and drug discovery.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Binding Sites
  • Hydrogen Bonding
  • Ligands
  • Proteins / chemistry*
  • Software*

Substances

  • Ligands
  • Proteins