Neuropeptide-S evoked arousal with electroencephalogram slow-wave compensatory drive in rats

Neuropsychobiology. 2012 Jun;65(4):195-205. doi: 10.1159/000336998. Epub 2012 Apr 26.

Abstract

Objectives: Neuropeptide S (NPS) exerts a dual arousal and anxiolytic effect in rodents, which may indicate the potential of a novel class of therapeutic agents in psychiatry. The purpose of this study is to fully describe the nature of electroencephalogram (EEG)-defined waking that mediates these arousal effects.

Methods: Effects of the intracerebroventricular infusion of NPS at 2 different doses were characterized over 20 h on sleep-wake architecture and EEG spectral components in rats that were chronically implanted with epidural electrodes for continuous measurement of sleep polygraphic and EEG variables.

Results: NPS (1 and 10 nmol) increased active waking (+88 and +87%, respectively), decreased light slow-wave sleep (lSWS) (-84 and -68%, respectively), deep slow-wave sleep (dSWS) (-47 and -33%, respectively) and rapid-eye-movement sleep (-71 and -70%, respectively) during the first 2 h after infusion. The wake-promoting effect of NPS is consistent with a marked lengthening in latency to sleep onset, a decrease in the number of state transitions from wakefulness to lSWS, and a delayed lSWS compensatory response. Interestingly, NPS significantly enhanced waking EEG theta oscillations and slow wave activity during dSWS.

Conclusion: The findings suggest that NPS enhanced a consolidated waking associated with a subsequent compensatory EEG slow-wave homeostatic drive rather than rebound sleep duration. The characteristics of NPS-induced waking coupled with enhanced EEG theta oscillations without rebound in sleep are desirable therapeutic features in wake-promoting agents.

MeSH terms

  • Animals
  • Arousal / drug effects*
  • Brain Waves / drug effects*
  • Dose-Response Relationship, Drug
  • Drive*
  • Electroencephalography
  • Eye Movements / drug effects
  • Eye Movements / physiology
  • Homeostasis / drug effects
  • Homeostasis / physiology
  • Male
  • Neuropeptides / pharmacology*
  • Polysomnography
  • Rats
  • Rats, Sprague-Dawley
  • Reaction Time / drug effects
  • Sleep Stages / drug effects
  • Statistics, Nonparametric
  • Wakefulness / drug effects

Substances

  • Neuropeptides
  • neuropeptide S, rat