Molecular evidence of curcumin-induced apoptosis in the filarial worm Setaria cervi

Parasitol Res. 2012 Sep;111(3):1173-86. doi: 10.1007/s00436-012-2948-0. Epub 2012 May 5.

Abstract

Curcumin (diferuloyl methane) is a major curcuminoid from Curcuma longa that exhibits various pharmacological effects and has shown multiple beneficial activities. Our understanding of its anticarcinogenic and other activities occurring through curcumin-induced apoptosis in several cancer cells has greatly expanded in recent years. Lymphatic filariasis is a worldwide health problem causing global disability in humans and is caused by filarial nematodes. Development of efficient strategies to promote programmed cell death in filarial worms remains a key challenge for anti-filarial drug developing research and a crucial unmet medical need. In this study, we have taken molecular and biochemical approaches toward understanding the molecular basis for curcumin-mediated anti-filarial activity in the filarial nematode Setaria cervi. Results of MTT assay showed that curcumin causes a significant reduction in viability of Mf and adults and thus acts as a potent macro- and micro-filaricidal agent. Hoechst staining, TUNEL staining, showed several apoptotic nuclei in different parts of curcumin-treated adults. At 25 μM concentration it showed chromosomal DNA fragmentation in adult worms. Our results indicate that curcumin decreases protein and mRNA expression levels of anti-apoptotic gene ced-9 and enhances both the levels of pro-apoptotic genes ced-3 and ced-4 in a dose-dependent manner. All these observations ascertained the apoptogenicity of curcumin at a minimum concentration of 50 μM in this filarial worm. Furthermore, we showed that curcumin causes depletion of parasitic glutathione level, enhances the activities of glutathione S-transferase and superoxide dismutase and stimulates rapid generation of reactive oxygen species (ROS). Here, we present molecular evidence on curcumin-induced apoptosis in the filarial nematode S. cervi with probable involvement of ROS in a caspase-dependent manner.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis / drug effects*
  • Benzimidazoles
  • Curcumin / pharmacology*
  • DNA, Complementary / chemical synthesis
  • DNA, Helminth
  • Female
  • In Situ Nick-End Labeling
  • Male
  • Nematoda / drug effects*
  • Oxidative Stress
  • RNA, Helminth
  • Reactive Oxygen Species
  • Staining and Labeling

Substances

  • Benzimidazoles
  • DNA, Complementary
  • DNA, Helminth
  • RNA, Helminth
  • Reactive Oxygen Species
  • Curcumin
  • bisbenzimide ethoxide trihydrochloride