Melanocortin-3 receptor regulates the normal fasting response

Proc Natl Acad Sci U S A. 2012 Jun 5;109(23):E1489-98. doi: 10.1073/pnas.1201994109. Epub 2012 May 9.

Abstract

The melanocortin-3 receptor-deficient (MC3-R(-/-)) mouse exhibits mild obesity without hyperphagia or hypometabolism. MC3-R deletion is reported to increase adiposity, reduce lean mass and white adipose tissue inflammation, and increase sensitivity to salt-induced hypertension. We show here that the MC3-R(-/-) mouse exhibits defective fasting-induced white adipose tissue lipolysis, fasting-induced liver triglyceride accumulation, fasting-induced refeeding, and fasting-induced regulation of the adipostatic and hypothalamic-adrenal-pituitary axes. Close examination of the hypothalamic-pituitary-adrenal axis showed that MC3-R(-/-) mice exhibit elevated nadir corticosterone as well as a blunted fasting-induced activation of the axis. The previously described phenotypes of this animal and the reduced bone density reported here parallel those of Cushing syndrome. Thus, MC3-R is required for communicating nutritional status to both central and peripheral tissues involved in nutrient partitioning, and this defect explains much of the metabolic phenotype in the model.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Absorptiometry, Photon
  • Adipose Tissue, White / metabolism
  • Adiposity / genetics
  • Adrenal Glands / cytology
  • Analysis of Variance
  • Animals
  • Biomechanical Phenomena
  • Blotting, Western
  • Body Composition / physiology
  • Corticosterone / metabolism
  • Energy Metabolism / physiology*
  • Fasting / physiology*
  • Hypothalamo-Hypophyseal System / physiology*
  • Immunohistochemistry
  • In Situ Hybridization
  • Lipolysis / physiology
  • Liver / metabolism
  • Male
  • Mice
  • Mice, Knockout
  • Pituitary-Adrenal System / physiology*
  • Real-Time Polymerase Chain Reaction
  • Receptor, Melanocortin, Type 3 / deficiency
  • Receptor, Melanocortin, Type 3 / physiology*
  • Triglycerides / metabolism

Substances

  • Receptor, Melanocortin, Type 3
  • Triglycerides
  • Corticosterone