A robust, high-sensitivity stealth probe for peptidases

Chem Commun (Camb). 2012 Jun 25;48(50):6253-5. doi: 10.1039/c2cc32227g. Epub 2012 May 18.

Abstract

A robust, modular fluorogenic probe system has been developed which allows the highly sensitive off-ON detection of aminopeptidase activity by releasing an exceptionally photostable, insoluble, phenolic ESIPT fluorophore. The probes generate no false positive signal in over 24 hours, but when activated give a signal within 10 minutes.

MeSH terms

  • Fluorescein / chemical synthesis
  • Fluorescein / chemistry*
  • Fluorescent Dyes / chemical synthesis
  • Fluorescent Dyes / chemistry*
  • Molecular Structure
  • Peptide Hydrolases / analysis*
  • Peptide Hydrolases / metabolism

Substances

  • Fluorescent Dyes
  • Peptide Hydrolases
  • Fluorescein